Sfoglia per Autore
Investigation of the interaction between the atypical agonist c[YpwFG] and MOR
2008-01-01 Gentilucci, Luca; Squassabia, Federico; De Marco, Rossella; Artali, Roberto; Cardillo, Giuliana; Tolomelli, Alessandra; Spampinato, Santi; Bedini, Andrea
Synthesis and conformational analysis of cyclotetrapeptide mimetic β-turn templates and validation as 3D scaffolds
2009-01-01 Gentilucci, L.; Cardillo, G.; Tolomelll, A.; De Marco, R.; Garelli, A.; Spampinato, S.; Sparta, A.; Juaristi, E.
Cyclopeptide analogs for generating new molecular and 3D diversity
2009-01-01 Gentilucci, L.; Cardillo, G.; Tolomelli, A.; Squassabia, F.; De Marco, R.; Chiriano, G.
Antiangiogenic effect of dual/selective α5 β1/αvβ3 integrin antagonists designed on partially modified retro-inverso cyclotetrapeptide mimetics
2010-01-01 Gentilucci, L.; Cardillo, G.; Spampinato, S.; Tolomelli, A.; Squassabia, F.; De Marco, R.; Bedini, A.; Baiula, M.; Belvisi, L.; Civera, M.
Chemical modifications designed to improve peptide stability: Incorporation of non-natural amino acids, pseudo-peptide bonds, and cyclization
2010-01-01 Gentilucci, L.; de Marco, R.; Cerisoli, L.
Peripheral antinociceptive effects of the cyclic endomorphin-1 analog c[YpwFG] in a mouse visceral pain model
2010-01-01 Bedini, A.; Baiula, M.; Gentilucci, L.; Tolomelli, A.; De Marco, R.; Spampinato, S.
The inverse type II β-Turn on D-Trp-Phe, a Pharmacophoric Motif for MOR Agonists
2011-01-01 Gentilucci, L.; Tolomelli, A.; de Marco, R.; Spampinato, S.; Bedini, A.; Artali, R.
Opioid activity profiles of oversimplified peptides lacking in the protonable N-terminus
2012-01-01 De Marco, R.; Tolomelli, A.; Spampinato, S.; Bedini, A.; Gentilucci, L.
Expedient synthesis of pseudo-Pro-containing peptides: Towards constrained peptidomimetics and foldamers
2012-01-01 De Marco, R.; Tolomelli, A.; Campitiello, M.; Rubini, P.; Gentilucci, L.
In-peptide synthesis of di-oxazolidinone and dehydroamino acid-oxazolidinone motifs as β-turn inducers
2013-01-01 De Marco, R.; Greco, A.; Rupiani, S.; Tolomelli, A.; Tomasini, C.; Pieraccini, S.; Gentilucci, L.
Cyclic side-chain-linked opioid analogs utilizing cis- and trans-4-aminocyclohexyl-d-alanine
2014-01-01 Piekielna, J.; Gentilucci, L.; De Marco, R.; Perlikowska, R.; Adamska, A.; Olczak, J.; Mazur, M.; Artali, R.; Modranka, J.; Janecki, T.; Tomboly, C.; Janecka, A.
Easy preparation of dehydroalanine building blocks equipped with oxazolidin-2-one chiral auxiliaries, and applications to the stereoselective synthesis of substituted tryptophans
2014-01-01 De Marco, R.; Cavina, L.; Greco, A.; Gentilucci, L.
Synthesis and assay of retro-α4β1 integrin-targeting motifs
2014-01-01 Dattoli, S. D.; De Marco, R.; Baiula, M.; Spampinato, S.; Greco, A.; Tolomelli, A.; Gentilucci, L.
Synthesis and Analysis of the Conformational Preferences of 5-Aminomethyloxazolidine-2,4-dione Scaffolds: First Examples of β2- and β2, 2-Homo-Freidinger Lactam Analogues
2014-01-01 Greco, A.; Tani, S.; De Marco, R.; Gentilucci, L.
Synthesis of tripeptides containing d-Trp substituted at the indole ring, assessment of opioid receptor binding and in vivo central antinociception
2014-01-01 De Marco, R.; Bedini, A.; Spampinato, S.; Gentilucci, L.
Diagnostic implementation of fast and selective integrin-mediated adhesion of cancer cells on functionalized zeolite L monolayers
2015-01-01 Greco, A.; Maggini, L.; De Cola, L.; De Marco, R.; Gentilucci, L.
Strategies to Improve Bioavailability and In Vivo Efficacy of the Endogenous Opioid Peptides Endomorphin-1 and Endomorphin-2
2015-01-01 De Marco, R; Janecka, A
5-aminomethyloxazolidine-2,4-dione hybrid α/β-dipeptide scaffolds as inductors of constrained conformations: Applications to the synthesis of integrin antagonists
2015-01-01 De Marco, R.; Mazzotti, G.; Dattoli, S. D.; Baiula, M.; Spampinato, S.; Greco, A.; Gentilucci, L.
Integrin Ligands with α/β-Hybrid Peptide Structure: Design, Bioactivity, and Conformational Aspects
2016-01-01 De Marco, R.; Tolomelli, A.; Juaristi, E.; Gentilucci, L.
Synthesis of mixed MOR/KOR efficacy cyclic opioid peptide analogs with antinociceptive activity after systemic administration
2016-01-01 Perlikowska, R.; Piekielna, J.; Gentilucci, L.; De Marco, R.; Cerlesi, M. C.; Calo, G.; Artali, R.; Tomboly, C.; Kluczyk, A.; Janecka, A.
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