Sfoglia per Autore
Investigation of the interaction between the atypical agonist c[YpwFG] and MOR
2008-01-01 Gentilucci, Luca; Squassabia, Federico; De Marco, Rossella; Artali, Roberto; Cardillo, Giuliana; Tolomelli, Alessandra; Spampinato, Santi; Bedini, Andrea
Synthesis and conformational analysis of cyclotetrapeptide mimetic β-turn templates and validation as 3D scaffolds
2009-01-01 Gentilucci, L.; Cardillo, G.; Tolomelll, A.; De Marco, R.; Garelli, A.; Spampinato, S.; Sparta, A.; Juaristi, E.
Cyclopeptide analogs for generating new molecular and 3D diversity
2009-01-01 Gentilucci, L.; Cardillo, G.; Tolomelli, A.; Squassabia, F.; De Marco, R.; Chiriano, G.
Peripheral antinociceptive effects of the cyclic endomorphin-1 analog c[YpwFG] in a mouse visceral pain model
2010-01-01 Bedini, A.; Baiula, M.; Gentilucci, L.; Tolomelli, A.; De Marco, R.; Spampinato, S.
Chemical modifications designed to improve peptide stability: Incorporation of non-natural amino acids, pseudo-peptide bonds, and cyclization
2010-01-01 Gentilucci, L.; de Marco, R.; Cerisoli, L.
Antiangiogenic effect of dual/selective α5 β1/αvβ3 integrin antagonists designed on partially modified retro-inverso cyclotetrapeptide mimetics
2010-01-01 Gentilucci, L.; Cardillo, G.; Spampinato, S.; Tolomelli, A.; Squassabia, F.; De Marco, R.; Bedini, A.; Baiula, M.; Belvisi, L.; Civera, M.
The inverse type II β-Turn on D-Trp-Phe, a Pharmacophoric Motif for MOR Agonists
2011-01-01 Gentilucci, L.; Tolomelli, A.; de Marco, R.; Spampinato, S.; Bedini, A.; Artali, R.
Expedient synthesis of pseudo-Pro-containing peptides: Towards constrained peptidomimetics and foldamers
2012-01-01 De Marco, R.; Tolomelli, A.; Campitiello, M.; Rubini, P.; Gentilucci, L.
Opioid activity profiles of oversimplified peptides lacking in the protonable N-terminus
2012-01-01 De Marco, R.; Tolomelli, A.; Spampinato, S.; Bedini, A.; Gentilucci, L.
In-peptide synthesis of di-oxazolidinone and dehydroamino acid-oxazolidinone motifs as β-turn inducers
2013-01-01 De Marco, R.; Greco, A.; Rupiani, S.; Tolomelli, A.; Tomasini, C.; Pieraccini, S.; Gentilucci, L.
Cyclic side-chain-linked opioid analogs utilizing cis- and trans-4-aminocyclohexyl-d-alanine
2014-01-01 Piekielna, J.; Gentilucci, L.; De Marco, R.; Perlikowska, R.; Adamska, A.; Olczak, J.; Mazur, M.; Artali, R.; Modranka, J.; Janecki, T.; Tomboly, C.; Janecka, A.
Easy preparation of dehydroalanine building blocks equipped with oxazolidin-2-one chiral auxiliaries, and applications to the stereoselective synthesis of substituted tryptophans
2014-01-01 De Marco, R.; Cavina, L.; Greco, A.; Gentilucci, L.
Synthesis of tripeptides containing d-Trp substituted at the indole ring, assessment of opioid receptor binding and in vivo central antinociception
2014-01-01 De Marco, R.; Bedini, A.; Spampinato, S.; Gentilucci, L.
Synthesis and Analysis of the Conformational Preferences of 5-Aminomethyloxazolidine-2,4-dione Scaffolds: First Examples of β2- and β2, 2-Homo-Freidinger Lactam Analogues
2014-01-01 Greco, A.; Tani, S.; De Marco, R.; Gentilucci, L.
Synthesis and assay of retro-α4β1 integrin-targeting motifs
2014-01-01 Dattoli, S. D.; De Marco, R.; Baiula, M.; Spampinato, S.; Greco, A.; Tolomelli, A.; Gentilucci, L.
Diagnostic implementation of fast and selective integrin-mediated adhesion of cancer cells on functionalized zeolite L monolayers
2015-01-01 Greco, A.; Maggini, L.; De Cola, L.; De Marco, R.; Gentilucci, L.
Strategies to Improve Bioavailability and In Vivo Efficacy of the Endogenous Opioid Peptides Endomorphin-1 and Endomorphin-2
2015-01-01 De Marco, R; Janecka, A
5-aminomethyloxazolidine-2,4-dione hybrid α/β-dipeptide scaffolds as inductors of constrained conformations: Applications to the synthesis of integrin antagonists
2015-01-01 De Marco, R.; Mazzotti, G.; Dattoli, S. D.; Baiula, M.; Spampinato, S.; Greco, A.; Gentilucci, L.
Integrin Ligands with α/β-Hybrid Peptide Structure: Design, Bioactivity, and Conformational Aspects
2016-01-01 De Marco, R.; Tolomelli, A.; Juaristi, E.; Gentilucci, L.
Synthesis of mixed MOR/KOR efficacy cyclic opioid peptide analogs with antinociceptive activity after systemic administration
2016-01-01 Perlikowska, R.; Piekielna, J.; Gentilucci, L.; De Marco, R.; Cerlesi, M. C.; Calo, G.; Artali, R.; Tomboly, C.; Kluczyk, A.; Janecka, A.
Heterocyclic Scaffolds in the Design of Peptidomimetic Integrin Ligands: Synthetic Strategies, Structural Aspects, and Biological Activity
2016-01-01 De Marco, R; Mazzotti, G; Greco, A; Gentilucci, L
Versatile Picklocks to Access All Opioid Receptors: Tuning the Selectivity and Functional Profile of the Cyclotetrapeptide c[Phe- d -Pro-Phe-Trp] (CJ-15,208)
2016-01-01 De Marco, R.; Bedini, A.; Spampinato, S.; Cavina, L.; Pirazzoli, E.; Gentilucci, L.
Modern tools for the chemical ligation and synthesis of modified peptides and proteins
2016-01-01 Gentilucci, L.; Tosi, P.; Bauer, A.; De Marco, R.
Redoubling the ring size of an endomorphin-2 analog transforms a centrally acting mu-opioid receptor agonist into a pure peripheral analgesic
2016-01-01 Piekielna, J.; De Marco, R.; Gentilucci, L.; Cerlesi, M. C.; Calo', G.; Tomboly, C.; Artali, R.; Janecka, A.
Tryptophan-Containing Non-Cationizable Opioid Peptides - A new chemotype with unusual structure and in vivo activity
2017-01-01 De Marco, R.; Gentilucci, L.
Design and characterization of opioid ligands based on cycle-in-macrocycle scaffold
2017-01-01 Adamska-Bartlomiejczyk, A.; De Marco, R.; Gentilucci, L.; Kluczyk, A.; Janecka, A.
Selective detection of α4β1 integrin (VLA-4)-expressing cells using peptide-functionalized nanostructured materials mimicking endothelial surfaces adjacent to inflammatory sites
2017-01-01 De Marco, R.; Greco, A.; Calonghi, N.; Dattoli, S. D.; Baiula, M.; Spampinato, S.; Picchetti, P.; De Cola, L.; Anselmi, M.; Cipriani, F.; Gentilucci, L.
. DS-70, a novel and potent 4 integrin antagonist, is an effective treatment for experimental allergic conjunctivitis in guinea pigs
2018-01-01 Deianira Dattoli, Samantha; Baiula, Monica; DE MARCO, Rossella; Bedini, Andrea; Anselmi, Michele; Gentilucci, Luca; Spampinato, Santi
Constraining Endomorphin-1 by β,α-Hybrid Dipeptide/Heterocycle Scaffolds: Identification of a Novel κ-Opioid Receptor Selective Partial Agonist
2018-01-01 De Marco, R.; Bedini, A.; Spampinato, S.; Comellini, L.; Zhao, J.; Artali, R.; Gentilucci, L.
In-Peptide Synthesis of Imidazolidin-2-one Scaffolds, Equippable with Proteinogenic or Taggable/Linkable Side Chains, General Promoters of Unusual Secondary Structures
2019-01-01 DE MARCO, Rossella; Zhao, J.; Greco, A.; Ioannone, S.; Gentilucci, L.
Stimuli-responsive local drug molecule delivery to adhered cells in a 3D nanocomposite scaffold
2019-01-01 Motealleh, A.; De Marco, R.; Kehr, N. S.
Integrin-Targeting Dye-Doped PEG-Shell/Silica-Core Nanoparticles Mimicking the Proapoptotic Smac/DIABLO Protein
2020-01-01 De Marco, R; Rampazzo, E; Zhao, J; Prodi, L; Paolillo, M; Picchetti, P; Gallo, F; Calonghi, N; Gentilucci, L
Functional Selectivity and Antinociceptive Effects of a Novel KOPr Agonist
2020-01-01 Bedini, A.; Di Cesare Mannelli, L.; Micheli, L.; Baiula, M.; Vaca, G.; De Marco, R.; Gentilucci, L.; Ghelardini, C.; Spampinato, S.
15N-Urea release evaluation from two types of mesoporous silica nanoparticles: perspectives for future application as slow release nanofertilizer
2021-01-01 Fellet, Guido; DE MARCO, Rossella; Pilotto, Laura; Marchiol, Luca
APE1 interacts with the nuclear exosome complex protein MTR4 and is involved in cisplatin- and 5-fluorouracil-induced RNA damage response
2022-01-01 Codrich, M.; Degrassi, M.; Malfatti, M. C.; Antoniali, G.; Gorassini, A.; Ayyildiz, D.; Marco, De; Giancarlo, Verardo; Tell, Gianluca
Editorial: Integrin Ligands and Their Bioconjugate Systems: Synthesis, Conformation, and Biological Activity
2022-01-01 De Marco, Rossella; Dehshahri, Ali; Baiula, Monica; Dodero, Veronica I.
High production of secondary metabolites and biological activities of Cydonia oblonga Mill. pulp fruit callus
2022-01-01 De Bellis, Roberta; Chiarantini, Laura; Potenza, Lucia; Gorassini, Andrea; Verardo, Giancarlo; De Marco, Rossella; Benayada, Leila; Stocchi, Vilberto; Cristina Albertini, Maria; Fraternale, Daniele
Dual-targeting peptides@PMO, a mimetic to the pro-apoptotic protein Smac/DIABLO for selective activation of apoptosis in cancer cells
2023-01-01 Di Giorgio, E.; Ferino, A.; Huang, W.; Simonetti, S.; Xodo, L.; De Marco, R.
POM@PMO plastic electrode for phosphate electrochemical detection: a further improvement of the detection limit
2023-01-01 Ben-Aissa, S.; De Marco, R.; Susmel, S.
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